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بنزيل فينتانيل

Benzylfentanyl (R-4129) is a fentanyl analog. It was temporarily placed in the US Schedule I by emergency scheduling in 1985 due to concerns about its potential for abuse as a designer drug, but this placement was allowed to expire and benzylfentanyl was formally removed from controlled substance listing in 2010, after the DEA's testing determined it to be "essentially inactive" as an opioid. It was added as a List I precursor instead in 2020 after it was determined that it was being used in fentanyl manufacture, which was previously thought to be beyond the technical capability of illicit labs. Benzylfentanyl has a Ki of 213 nM at the mu opioid receptor, binding around ⁠1/200⁠ as strong as fentanyl itself, though it is still slightly more potent than codeine.

بنزيل فينتانيل molecular structure
بنزيل فينتانيل molecular structure diagram from the DrugsPRO substance library.

Classification

  • Chemical: Anilidopiperidine
  • Chemical: Opioid
  • Psychoactive: Depressant

Effects

  • Sedation
  • Motor Impairment
  • Respiratory Depression
  • Constipation
  • Pupil Constriction
  • Itchiness
  • Reduced Anxiety
  • Euphoria
  • Anxiety Suppression
  • Dulled Perception

Routes of Administration

No route information available yet.

Harm Reduction

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Sources

Substance data is aggregated from the following public harm-reduction and reference sources.

Links

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Benzylfentanyl - دليل المواد DrugsPRO

Benzylfentanyl: Benzylfentanyl (R-4129) is a fentanyl analog. It was temporarily placed in the US Schedule I by emergency scheduling in 1985 due to concerns about its potential for abuse as a designer drug, but this placement was allowed to expire and benzylfentanyl was formally removed from control

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